用于肿瘤及相关领域研究的生物活性化合物。
Favipiravir, also known as T-705 or Avigan, is an experimental antiviral drug being developed by Toyama Chemical of...
FGFR3-IN-10 is a FGFR3 inhibitor with superior selectivity for FGFR3 over FGFR1 .FGFR3-IN-10 can be used for the...
KRAS G12C inhibitor 41 is a potent inhibitor of KRAS G12C . The Ras family of proteins is an important intracellular...
Acalabrutinib, also known as ACP-196, is an orally available inhibitor of Bruton's tyrosine kinase (BTK) with...
PDGFRα kinase inhibitor 2 (compound 1), an Imatinib ( HY-15463 ) analogue, is a covalent and irreversible kinase...
FASN-IN-3 is a fatty acid synthase ( FASN ) inhibitor extracted from patent US20170119786A1, compound 242A.
AZD-0284 is a selective inverse agonist of the nuclear receptor RORγ . AZD-0284 has the potential for plaque...
CDK7-IN-1, an analog of YKL-5-124, is a cyclin-dependent kinase 7 ( cdk7 ) inhibitor, with an IC 50 of less than 100...
Tivozanib is an orally bioavailable inhibitor of vascular endothelial growth factor receptors (VEGFRs) 1, 2 and 3...
JR4-187 is an orally active, copper-dependent anticancer agent. JR4-187 downregulates genes involved in oxidative...
golvatinib (also known as E7050) is an orally bioavailable dual kinase inhibitor of c-Met (hepatocyte growth factor...
VAL-083 is a bi-functional alkylating agent that inhibits U251 and SF188 cell growth in monolayer better than TMZ...
BGG463 (K03859) is an orally active type II CDK2 inhibitor.
ATM-IN-13 (A36) is an orally active, selective ATM kinase inhibitor with a human IC 50 of 0.3 nM. ATM-IN-13 blocks...
PK11000 is an alkylating agent, and stabilizes the DNA-binding domain of both WT and mutant p53 proteins by covalent...
Glycycoumarin is a potent antispasmodic agent. Glycycoumarin is a major bioactive coumarin of licorice and exhibits...
Glucoraphanin, a natural glucosinolate found in cruciferous vegetable, is a stable precursor of the Nrf2 inducer...
CUR5g is a potent autophagy inhibitor. CUR5g selectively inhibits autophagosome degradation in cancer cells by...
KDM5A-IN-1 is a potent, orally bioavailable pan- histone lysine demethylases 5 ( KDM5 ) inhibitor with IC 50 s of 45...
KRP-203 monophosphate is a monophosphate of KRP-203 ( HY-13660 ). KRP-203 is an orally active...
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