(3aS,4R,9bR)-G-1

Overview

(3aS,4R,9bR)-G-1 is a highly selective G protein-coupled receptor GPR30 ( GPER ) agonist with a K i value of approximately 7 nM. (3aS,4R,9bR)-G-1 activates rapid signaling pathways such as intracellular calcium mobilization and PI3K signaling through GPR30, promoting uterine epithelial cell proliferation and exerting antidepressant effects. (3aS,4R,9bR)-G-1 is promising for research of breast cancer and depression.

Application

Products | Products > Disease Areas > Neurological, Eye or Ear Disease | Products > Signaling Pathways > GPCR/G Protein | Products > Signaling Pathways > PI3K/Akt/mTOR | Products > Research Areas > Cancer > Cancer Metabolism and Metastasis | Products > Research Areas > Neurological Disease | Products > Research Areas > Cancer | Products > Research Areas > Cancer > Cancer Targeted Therapy | Products > Signaling Pathways > Adhesion G Protein-coupled Receptors (AGPCRs) | Products > Signaling Pathways > PI3K

Product Information

• Catalog No.: HY-107216A
• CAS No.: 925419-53-0
• Molecular Formula: C21H18BrNO3
• Molecular Weight: 412.28
• Purity: 99.98%
• Storage: Please store the product under the recommended conditions in the Certificate of Analysis.

Source

Original product source