FR 180204

Overview

FR 180204 is an ATP-competitive and selective ERK inhibitor. FR 180204 inhibits ERK1 and ERK2 with IC 50 s of 0.51 μM ( K i =0.31 μM) and 0.33 μM ( K i =0.14 μM), respectively.

Application

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Product Information

• Catalog No.: HY-12275
• CAS No.: 865362-74-9
• Molecular Formula: C18H13N7
• Molecular Weight: 327.34
• Purity: 99.91%
• Storage: Powder -20°C, 3 years , 4°C, 2 years ; In solvent -80°C, 2 years , -20°C, 1 year
• Solubility: ≥ 2.5 mg/mL (7.64 mM); Clear solution
• Availability: In-stock

Source

Original product source