GSK163090

Overview

GSK163090 is a potent, selective and orally active 5-HT 1A/1B/1D receptor antagonist with pK i values of 9.4, 8.5 and 9.7, respectively. GSK163090 inhibits the functional activity of serotonin reuptake transporter (SerT) with a pK i value of 6.1. GSK163090 has antidepressant and anxiolytic activities.

Application

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Product Information

• Catalog No.: HY-14348
• CAS No.: 844903-58-8
• Molecular Formula: C25H29N5O
• Molecular Weight: 415.53
• Purity: 99.57%
• Storage: Powder -20°C, 3 years , 4°C, 2 years ; In solvent -80°C, 2 years , -20°C, 1 year
• Solubility: ≥ 1.43 mg/mL (3.44 mM); Clear solution
• Availability: In-stock

Source

Original product source