Levomilnacipran-d 10 hydrochloride

Overview

Levomilnacipran-d 10 ((1S,2R)-Milnacipran-d 10 ) hydrochloride is deuterium labeled Levomilnacipran hydrochloride ( HY-B0168B ). Levomilnacipran ((1S,2R)-Milnacipran) hydrochloride is the enantiomer of Milnacipran ( HY-B0168 ) and a strong substrate of P-gp that can cross the blood-brain barrier. Levomilnacipran hydrochloride is a serotonin and norepinephrine reuptake inhibitor, with IC 50 values of 10.5 nM and 19.0 nM, and K i values of 92.2 nM and 1.2 nM for human norepinephrine transporter ( NET ) and serotonin transporter ( SERT ), respectively. Levomilnacipran hydrochloride has antidepressant and anxiolytic activities. Levomilnacipran hydrochloride can be used for the research of depression.

Application

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Product Information

• Catalog No.: HY-14794AS
• CAS No.: 2747914-23-2
• Molecular Formula: C15H13D10ClN2O
• Molecular Weight: 292.87
• Purity: 99.98%
• Storage: Please store the product under the recommended conditions in the Certificate of Analysis.

Source

Original product source