L-838417-d 9

Overview

L-838417 -d 9 is the deuterium labeled L-838417 ( HY-W009009 ). L-838417 is a selective partial agonist at the α2, α3 and α5 subtypes of the GABA A receptor and an antagonist at the α1, with binding K i values of 0.79 nM, 0.67 nM, 1.67 nM, 267 nM, 2.25 nM and 2183 nM for α1β3γ2, α2β3γ2, α3β3γ2, α4β3γ2, α5β3γ2 and α6β3γ2. L-838417 has anti-anxiety activity.

Application

Products | Products > Disease Areas > Neurological, Eye or Ear Disease | Products > Signaling Pathways > Others | Products > Signaling Pathways > Membrane Transporter/Ion Channel | Products > Signaling Pathways > Neuronal Signaling | Products > Research Areas > Neurological Disease | Products > Signaling Pathways > Isotope-Labeled Compounds | Products > Signaling Pathways > GABA Receptor

Product Information

• Catalog No.: HY-15831
• CAS No.: 1213669-91-0
• Molecular Formula: C19H10D9F2N7O
• Molecular Weight: 408.45
• Purity: 99.74%
• Storage: Powder -20°C, 3 years ; In solvent -80°C, 6 months , -20°C, 1 month
• Availability: In-stock

Source

Original product source