Plazomicin (ACHN 490) is a semi-synthetic aminoglycoside Antibiotic . Plazomicin acts as a substrate for Aminoglycoside acetyltransferase and Aminoglycoside phosphotransferase . Plazomicin is not modified by various common aminoglycoside-modifying enzymes . Plazomicin selectively inhibits MATE2-K . Plazomicin exhibits activity against multidrug-resistant bacteria, including carbapenem-resistant Enterobacterales.
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