Lumateperone-d 4

Overview

Lumateperone-d 4 (ITI-007-d 4 ) is deuterium labeled Lumateperone. Lumateperone (ITI-007) is an orally active 5-HT2A receptor antagonist (Ki = 0.54 nM), a partial agonist of presynaptic D2 receptors and an antagonist of postsynaptic D2 receptors (Ki = 32 nM), and a dopamine D1 receptor modulator. Lumateperone has anticancer activity and can also be used for the study of schizophrenia and bipolar depression.

Application

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Product Information

• Catalog No.: HY-17637S2
• CAS No.: 2102683-55-4
• Molecular Formula: C24H24D4FN3O
• Molecular Weight: 397.52
• Purity: 99.98%
• Storage: Please store the product under the recommended conditions in the Certificate of Analysis.

Source

Original product source