Ziptide is a substrate for MAPK activated protein kinase 2 ( MAPKAPK2 , K m = 5 μM), MAPKAPK3 (K m = 30 μM), PARK (K m = 40 μM), checkpoint kinase 1 ( Chk1 , K m = 5 μM), AMP-activated protein kinase ( AMPK , K m = 75 μM), and calcium/calmodulin-dependent protein kinase II (CamKII, K m = 300 μM).
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