(S)-(+)-Dimethindene maleate (Standard)

Overview

(S)-(+)-Dimethindene maleate (Standard) is the analytical standard of (S)-(+)-Dimethindene (maleate) ( HY-107647 ). This product is intended for research and analytical applications. (S)-(+)-Dimethindene maleate , an enantiomer, is a potent M2-selective muscarinic receptor antagonist (pA2 = 7.86/7.74; pK i = 7.78). (S)-(+)-Dimethindene maleate shows lower affinities for the muscarinic M1 (pA2 = 6.83/6.36; pK i = 7.08), the M3 (pA2 = 6.92/6.96; pK i = 6.70) and the M4 receptors (pK i = 7.00), respectively. (S)-(+)-Dimethindene maleate also is a histamine H1 receptor antagonist (pA2 = 7.48).

Application

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Product Information

• Catalog No.: HY-107647R
• CAS No.: 136152-65-3
• Molecular Formula: C24H28N2O4
• Molecular Weight: 408.49
• Storage: Please store the product under the recommended conditions in the Certificate of Analysis.

Source

Original product source