GSK-5959 CAS:901245-65-6 is a potent, selective and cell-permeable BRPF1 bromodomain inhibitor with IC50 ~80 nM. More than 100-fold selectivity for BRPF1 (IC50 = 80 nM) over other 35 bromodomains including BRPF2/3 and BET family bromodomains.
Polyethylene Glycol PEG Linkers > PROTAC Linker > BET Inhibitors
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