Other grades of this product :
| J104129 Basic information |
| J104129 Chemical Properties |
| storage temp. | 2-8°C | | form | powder | | color | white to beige | | optical activity | [α]/D -6 to -8°, c = 1 in methanol |
| J104129 Usage And Synthesis |
| Uses | J 104129 Fumarate is a novel muscarinic M3 receptor antagonist with high selectivity for M3 over M2 receptors. | | Biochem/physiol Actions | J104129 is a muscarinic M3 receptor antagonist greater than 100-fold selectivity for M3 over M2 receptors. Its Ki for M3 receptors = 4.2 nM compared to a Ki of 490 nM for M2 receptors. J-104129 showed potent bronchodilator activity in animal studies. |
| J104129 Preparation Products And Raw materials |
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