BLU-667

Overview

BLU-667 (Pralsetinib) is a highly effective and selective RET inhibitor. It has an IC50 of 0.3-0.4 nM for the fusion of WT RET, RET mutants V804L, V804M, M918T and CCDC6-RET.

Application

Products > Drug Discovery > Inhibitor > Other Inhibitors | Products > Drug Discovery > Inhibitor

Product Information

• Catalog No.: B2693-373106
• CAS No.: 2097132-94-8
• Molecular Formula: C27H32FN9O2
• Molecular Weight: 533.6
• Purity: ≥98% by HPLC
• Storage: Store at -20°C
• Solubility: Soluble in DMSO

Source

Original product source