Didesmethyl cariprazine (Standard)

Overview

Didesmethyl cariprazine (Standard) is the analytical standard of Didesmethyl cariprazine ( HY-100658 ). This product is intended for research and analytical applications. Didesmethyl cariprazine is an orally active, BBB-permeable metabolite of Cariprazine ( HY-14763 ). Didesmethyl cariprazine is a partial agonist at the D2 and D3 receptors, full agonist at the 5-HT1A receptor, and antagonist at the human 5-HT2B receptor (Ki: 1.41 nM (human D2L), 0.056 nM (human D3), 1.7 nM (human 5-HT1A), 0.52 nM (human 5-HT2B)). Didesmethyl cariprazine dose-dependently inhibits the spontaneous activity of rat midbrain dopaminergic neurons.

Application

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Product Information

• Catalog No.: HY-100658R
• CAS No.: 839712-25-3
• Molecular Formula: C19H28Cl2N4O
• Molecular Weight: 399.36
• Purity: 98%
• Storage: Please store the product under the recommended conditions in the Certificate of Analysis.
• Availability: In-stock

Source

Original product source