Silodosin

Overview

Silodosin (KAD 3213; KMD 3213) is a potent, selective and orally active α1A-adrenergic receptor (α1A-AR) blocker. Silodosin exhibits high affinity for α1A-AR ( K i =0.036 nM), over 162-fold and 50-fold than for α1B-AR and α1D-AR with K i values of 21 nM and 2.0 nM, respectively. Silodosin is an effective and well-tolerated agent, it can be used for the investigation of LUTS/BPH.

Application

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Product Information

• Catalog No.: HY-10122
• CAS No.: 160970-54-7
• Molecular Formula: C25H32F3N3O4
• Molecular Weight: 495.53
• Purity: 99.89%
• Storage: Powder -20°C, 3 years , 4°C, 2 years ; In solvent -80°C, 2 years , -20°C, 1 year
• Solubility: ≥ 2.5 mg/mL (5.05 mM); Clear solution
• Availability: In-stock

Source

Original product source