Conessine

Overview

Conessine is an orally active and BBB-penetrable selective histamine H3 receptor antagonist. The pK i values of Conessine for rat and human H3 receptors are 7.61 and 8.27, respectively. Conessine is an inhibitor of the multidrug efflux pump system in Pseudomonas aeruginosa and can enhance the activity of antibiotics . Conessine has antimalarial activity. Conessine can also be used in the research of muscle atrophy.

Application

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Product Information

• Catalog No.: HY-107566
• CAS No.: 546-06-5
• Molecular Formula: C24H40N2
• Molecular Weight: 356.59
• Purity: 99.87%
• Storage: -20°C, sealed storage, away from moisture and light * In solvent : -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture and light)
• Solubility: ≥ 2.5 mg/mL (7.01 mM); Clear solution
• Availability: In-stock

Source

Original product source