Momelotinib sulfate

Overview

Momelotinib sulfate (CYT387 sulfate salt) is an ATP-competitive inhibitor of JAK1/JAK2 with IC 50 of 11 nM/18 nM, 10-fold selectivity versus JAK3 (IC 50 =155 nM).

Application

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Product Information

• Catalog No.: HY-10962
• CAS No.: 1056636-06-6
• Molecular Formula: C23H26N6O10S2
• Molecular Weight: 610.62
• Purity: 98.45%
• Storage: -20°C, sealed storage, away from moisture * In solvent : -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture)
• Solubility: ≥ 3 mg/mL (4.91 mM); Clear solution
• Availability: In-stock

Source

Original product source