BI-671800

Overview

BI-671800 is a highly specific and potent antagonist of chemoattractant receptor-homologous molecule on Th2 cells (DP2/CRTH2) , with IC 50 values of 4.5 nM and 3.7 nM for PGD2 binding to CRTH2 in hCRTH2 and mCRTH2 transfected cells, respectively. BI-671800 has potential for the treatment of poorly controlled asthma.

Application

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Product Information

• Catalog No.: HY-114141
• CAS No.: 1093108-50-9
• Molecular Formula: C25H26F3N5O3
• Molecular Weight: 501.50
• Purity: 99.36%
• Storage: 4°C, protect from light * In solvent : -80°C, 6 months; -20°C, 1 month (protect from light)
• Solubility: ≥ 2.25 mg/mL (4.49 mM); Clear solution
• Availability: In-stock

Source

Original product source