BMS-986122

CAS No.：313669-88-4
Grade：99.90%
Formula：C16H15BrClNO3S2
M.W.：448.78
Solvent：2.5 mg/mL (5.57 mM); Suspended solution; Need ultrasonic

Important Notice

This product is a chemical product/pharmaceutical intermediate. It is not a drug, an active pharmaceutical ingredient (API), or a pharmaceutical-grade material. It has not been granted a drug approval number or a Chemical Drug Substance Approval Notice, has not passed drug-related review and approval, and is not manufactured, tested, or released in accordance with pharmaceutical GMP.
This product is intended solely for non-clinical research, process development, quality studies, further chemical processing, or chemical synthesis. It must not be used in drug-product manufacturing, clinical trials, clinical diagnosis, or administration to humans or animals, or be sold, used as an input, submitted for regulatory filing, or released as an API or pharmaceutical material.
The purchaser must not use this product, or supply it to another party, for personal consumption, sports or fitness, weight loss, health supplements, food, or animal feed.

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Overview

BMS-986122 is a selective, potent positive allosteric modulator of the mu-opioid receptor (µ-OR) . BMS-986122 shows potentiation of orthosteric agonist-mediated β-arrestin recruitment, adenylyl cyclase inhibition, and G protein activation. BMS-986122 potentiates DAMGO-mediated [ 35 S]GTPγS binding in mouse brain membranes.

Application

Product Information

Catalog No.: HY-120645
CAS No.: 313669-88-4
Molecular Formula: C16H15BrClNO3S2
Molecular Weight: 448.78
Purity: 99.90%
Storage: Powder -20°C, 3 years , 4°C, 2 years ; In solvent -80°C, 6 months , -20°C, 1 month
Solubility: 2.5 mg/mL (5.57 mM); Suspended solution; Need ultrasonic
Availability: In-stock

Source

Original product source

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