CP-99994 hydrochloride

Overview

CP-99994 hydrochloride is a Tachykinin neurokinin 1 (NK-1) receptor antagonist with a K i of 0.25 nM. CP-99994 hydrochloride prevents colorectal sensitization in the context of visceral hypersensitivity. CP-99994 hydrochloride reduces colorectal hypersensitivity induced by acetic acid injections in a model of bladder-colon cross-sensitization. CP-99994 hydrochloride attenuates the neuroglial interactions and MAPK-p38 phosphorylation associated with visceral hypersensitivity.

Application

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Product Information

• Catalog No.: HY-12145
• CAS No.: 145148-39-6
• Molecular Formula: C19H26Cl2N2O
• Molecular Weight: 369.33
• Purity: 99.98%
• Storage: Please store the product under the recommended conditions in the Certificate of Analysis.
• Availability: In-stock

Source

Original product source