BMS-819881

Overview

BMS-819881 is a melaninconcentrating hormone receptor 1 ( MCHR1 ) antagonist, which binds rat MCHR1 with a K i of 7 nM. BMS-819881 also is selective and potent for CYP3A4 activity with an EC 50 of 13 μM.

Application

Products | Products > Disease Areas > Metabolic or Endocrine Disease | Products > Signaling Pathways > GPCR/G Protein | Products > Signaling Pathways > Neuronal Signaling | Products > Signaling Pathways > Metabolic Enzyme/Protease | Products > Research Areas > Metabolic Disease | Products > Research Areas > Endocrinology | Products > Signaling Pathways > MCHR1 (GPR24) | Products > Signaling Pathways > Cytochrome P450

Product Information

• Catalog No.: HY-12433
• CAS No.: 1197420-05-5
• Molecular Formula: C24H21ClN2O4S
• Molecular Weight: 468.95
• Purity: 99.78%
• Storage: Powder -20°C, 3 years , 4°C, 2 years ; In solvent -80°C, 6 months , -20°C, 1 month
• Solubility: ≥ 2.5 mg/mL (5.33 mM); Clear solution
• Availability: In-stock

Source

Original product source