VU0810464

Overview

VU0810464 is a potent and selective non-ureaG protein-gated inwardly-rectifying potassium channels ( GIRK, Kir3 ) activator. VU0810464 displays nanomolar potency for neuronal ( EC 50 =165 nM) and GIRK1/4 ( EC 50 =720 nM) channels with improved brain penetration.

Application

Products | Products > Disease Areas > Neurological, Eye or Ear Disease | Products > Signaling Pathways > Membrane Transporter/Ion Channel | Products > Research Areas > Neurological Disease | Products > Signaling Pathways > Potassium Channel

Product Information

• Catalog No.: HY-127106
• CAS No.: 2126040-21-7
• Molecular Formula: C18H21ClFN3O
• Molecular Weight: 349.83
• Purity: 99.29%
• Storage: Powder -20°C, 3 years , 4°C, 2 years ; In solvent -80°C, 2 years , -20°C, 1 year
• Solubility: ≥ 2.08 mg/mL (5.95 mM); Clear solution
• Availability: In-stock

Source

Original product source