EHop-016

Overview

EHop-016 is a potent and selective Rac GTPase Rac1 and Rac3 inhibitor. EHop-016 inhibits Rac1 activity with an IC 50 of 1.1 μM in MDA-MB-435 cells. EHop-016 inhibits Vav2 interaction with Rac, Rac-activated PAK1 , lamellipodia formation, and cell migration.

Application

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Product Information

• Catalog No.: HY-12810
• CAS No.: 1380432-32-5
• Molecular Formula: C25H30N6O
• Molecular Weight: 430.55
• Purity: 99.38%
• Storage: Powder -20°C, 3 years , 4°C, 2 years ; In solvent -80°C, 2 years , -20°C, 1 year
• Solubility: ≥ 2.5 mg/mL (5.81 mM); Clear solution
• Availability: In-stock

Source

Original product source