KB-0742 dihydrochloride

Overview

KB-0742 dihydrochloride is a potent, selective and orally active CDK9 inhibitor with an IC 50 of 6 nM for CDK9/cyclin T1 . KB-0742 dihydrochloride is selective for CDK9/cyclin T1 with >50-fold selectivity over other CDK kinases. KB-0742 dihydrochloride has potent anti-tumor activity.

Application

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Product Information

• Catalog No.: HY-137478A
• CAS No.: 2416874-75-2
• Molecular Formula: C16H27Cl2N5
• Molecular Weight: 360.33
• Purity: 98.77%
• Storage: 4°C, sealed storage, away from moisture * In solvent : -80°C, 1 year; -20°C, 6 months (sealed storage, away from moisture)
• Solubility: ≥ 2.08 mg/mL (5.77 mM); Clear solution
• Availability: In-stock

Source

Original product source