α-NETA

Overview

α-NETA is a potent and noncompetitive choline acetyltransferase (ChA) inhibitor with an IC 50 of 9 μM. α-NETA is a potent ALDH1A1 ( IC 50 =0.04 µM) and chemokine-like receptor-1 (CMKLR1) antagonist. α-NETA weakly inhibits cholinesterase (ChE; IC 50 =84 µM) and acetylcholinesterase ( AChE ; IC 50 =300 µM). α-NETA has anti-cancer activity.

Application

Products | Products > Signaling Pathways > GPCR/G Protein | Products > Signaling Pathways > Metabolic Enzyme/Protease | Products > Signaling Pathways > Neuronal Signaling | Products > Signaling Pathways > Apoptosis | Products > Research Areas > Cancer | Products > Research Areas > Cancer > Cancer Targeted Therapy | Products > Research Areas > Cancer > Cancer Metabolism and Metastasis | Products > Signaling Pathways > Chemerin Receptor | Products > Signaling Pathways > Aldehyde Dehydrogenase (ALDH) | Products > Signaling Pathways > Cholinesterase (ChE) | Products > Signaling Pathways > Apoptosis

Product Information

• Catalog No.: HY-138097
• CAS No.: 115066-04-1
• Molecular Formula: C16H20INO
• Molecular Weight: 369.24
• Purity: ≥98.0%
• Storage: Powder -20°C, 3 years , 4°C, 2 years ; In solvent -80°C, 6 months , -20°C, 1 month
• Solubility: ≥ 2.08 mg/mL (5.63 mM); Clear solution
• Availability: In-stock

Source

Original product source