Palacaparib

Overview

AZD-9574 is a potent and brain penetrant PARP1 inhibitor and shows >8000-fold selectivity for PARP1 compared to PARP2/3/5a/6. AZD-9574 acts by selectively inhibiting and trapping PARP1 at the sites of SSBs. AZD-9574 is an anti-cancer agent and can be used for HRD + ?breast cancer and advanced solid malignancies research.

Application

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Product Information

• Catalog No.: HY-145804
• CAS No.: 2756333-39-6
• Molecular Formula: C21H22F2N6O2
• Molecular Weight: 428.44
• Purity: 98.30%
• Storage: Powder -20°C, 3 years , 4°C, 2 years ; In solvent -80°C, 6 months , -20°C, 1 month
• Solubility: ≥ 2.22 mg/mL (5.18 mM); Clear solution
• Availability: In-stock

Source

Original product source