PP487 is a selective dual inhibitor of Tyrosine kinase/PI3-K , with IC 50 values of 0.017 μM, 0.072 μM, 0.004 μM, 0.01 μM, 0.55 μM, 0.22 μM, and < 0.01 μM against DNA-PK , mTOR , Hck , Src , EGFR , EphB4 , and PDGFR , respectively. PP487 can be used in cancer research.
Products | Products > Disease Areas > Cancer | Products > Signaling Pathways > Protein Tyrosine Kinase/RTK | Products > Signaling Pathways > PI3K/Akt/mTOR | Products > Signaling Pathways > Cell Cycle/DNA Damage | Products > Signaling Pathways > JAK/STAT Signaling | Products > Research Areas > Cancer | Products > Research Areas > Cancer > Cancer Targeted Therapy | Products > Research Areas > Cancer > Cancer Metabolism and Metastasis | Products > Signaling Pathways > Bcr-Abl | Products > Signaling Pathways > Src | Products > Signaling Pathways > VEGFR | Products > Signaling Pathways > EGFR | Products > Signaling Pathways > PDGFR | Products > Signaling Pathways > c-Met/HGFR | Products > Signaling Pathways > PI3K | Products > Signaling Pathways > DNA-PK | Products > Signaling Pathways > mTOR
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