Relenopride hydrochloride

Overview

Relenopride (YKP10811) hydrochloride is a specific and selective 5-HT 4 receptor agonist ( K i =4.96 nM). Relenopride hydrochloride has 120-fold and 6-fold lower affinity, respectively, for 5-HT 2A (K i =600 nM) and 5-HT 2B receptors (K i =31 nM) than for 5-HT 4 . Relenopride hydrochloride increases gastrointestinal (GI) motility.

Application

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Product Information

• Catalog No.: HY-16729A
• CAS No.: 1221416-42-7
• Molecular Formula: C24H31Cl2FN4O4
• Molecular Weight: 529.43
• Purity: 99.85%
• Storage: -20°C, protect from light, stored under nitrogen * In solvent : -80°C, 6 months; -20°C, 1 month (protect from light, stored under nitrogen)
• Solubility: ≥ 2.75 mg/mL (5.19 mM); Clear solution
• Availability: In-stock

Source

Original product source