Gallamine

Overview

Gallamine is an allosteric, selective muscarinic M2 acetylcholine receptor antagonist ( EC 50 : 130 nM for [ 3 H]NMS dissociation from porcine muscarinic M2 receptors). Gallamine is also an acetylcholinesterase inhibitor ( IC 50 s : 1070 μM, 1480 μM, 235 μM for EeAChE, hAChE, hBChE, respectively (in the absence of MeCN)). Gallamine increases free norepinephrine levels. Gallamine can be used as a muscle relaxant.

Application

Products | Products > Disease Areas > Musculoskeletal and Skin Disease | Products > Signaling Pathways > GPCR/G Protein | Products > Signaling Pathways > Neuronal Signaling | Products > Research Areas > Inflammation/Immunology | Products > Signaling Pathways > mAChR | Products > Signaling Pathways > Cholinesterase (ChE)

Product Information

• Catalog No.: HY-180358
• CAS No.: 153-76-4
• Molecular Formula: C24H45N3O3
• Molecular Weight: 423.63
• Purity: 99.98%
• Storage: Please store the product under the recommended conditions in the Certificate of Analysis.

Source

Original product source