GSK864

Overview

GSK864, a chemical probe, is an isocitrate dehydrogenase 1 ( IDH1 ) mutant inhibitor; inhibits IDH1 mutants R132C, R132H, and R132G with IC 50 values of 8.8, 15.2 and 16.6 nM.

Application

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Product Information

• Catalog No.: HY-19540
• CAS No.: 1816331-66-4
• Molecular Formula: C30H31FN6O4
• Molecular Weight: 558.60
• Purity: 99.91%
• Storage: Powder -20°C, 3 years , 4°C, 2 years ; In solvent -80°C, 2 years , -20°C, 1 year
• Solubility: ≥ 2.5 mg/mL (4.48 mM); Clear solution
• Availability: In-stock

Source

Original product source