Isamoltane hemifumarate

Overview

Isamoltane hemifumarate is a selective antagonist of 5-HT 1B receptor , with an IC 50 of 39 nM for inhibits the binding of [ 125 I]ICYP to 5-HT 1B recognition sites in rat brain membranes. Isamoltane hemifumarate is also a β-adrenoceptor ligand, with an IC 50 of 8.4 nM. Isamoltane hemifumarate shows anxiolytic activity.

Application

Products | Products > Disease Areas > Neurological, Eye or Ear Disease | Products > Signaling Pathways > GPCR/G Protein | Products > Signaling Pathways > Neuronal Signaling | Products > Research Areas > Neurological Disease | Products > Signaling Pathways > 5-HT Receptor | Products > Signaling Pathways > Adrenergic Receptor

Product Information

• Catalog No.: HY-19578B
• CAS No.: 874882-92-5
• Molecular Formula: C16H22N2O2.1/2C4H4O4
• Molecular Weight: 332.40
• Purity: 99.98%
• Storage: Please store the product under the recommended conditions in the Certificate of Analysis.
• Availability: In-stock

Source

Original product source