Darifenacin

Overview

Darifenacin (UK-88525) is a selective and orally active M3 muscarinic receptor ( M3R ) antagonist with a pKi of 8.9. Darifenacin binds >20-fold more specifically to M3R than to other muscarinic receptors. Darifenacin can be used in the study of urinary incontinence and other symptoms of overactive bladder. Darifenacin inhibits tumor growth in colorectal cancer cells and has anti-tumor effects.

Application

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Product Information

• Catalog No.: HY-A0033
• CAS No.: 133099-04-4
• Molecular Formula: C28H30N2O2
• Molecular Weight: 426.55
• Purity: 99.81%
• Storage: Powder -20°C, 3 years , 4°C, 2 years ; In solvent -80°C, 6 months , -20°C, 1 month
• Solubility: 2.5 mg/mL (5.86 mM); Clear solution; Need ultrasonic
• Availability: In-stock

Source

Original product source