Desvenlafaxine

Overview

Desvenlafaxine, the succinate salt form of the isolated major active metabolite of Venlafaxine ( HY-B0196 ), is an orally active and BBB penetrated 5-HT and norepinephrine reuptake inhibitor, with IC 50 values of 47.3 nM and 531.3 nM for hSERT and hNET, respectively. Desvenlafaxine shows weak binding affinity (62% inhibition at 100 μM) at the human dopamine (DA) transporter.

Application

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Product Information

• Catalog No.: HY-B0602
• CAS No.: 93413-62-8
• Molecular Formula: C16H25NO2
• Molecular Weight: 263.38
• Purity: 99.76%
• Storage: Powder -20°C, 3 years , 4°C, 2 years ; In solvent -80°C, 6 months , -20°C, 1 month
• Solubility: ≥ 2.5 mg/mL (9.49 mM); Clear solution
• Availability: In-stock

Source

Original product source