Metergoline

Overview

Metergoline is a serotonin (5-HT) receptor and dopamine receptors antagonist, with pK i s of 8.64, 8.75 and 8.75 for 5-HT 2A , 5-HT 2B and 5-HT 2C , respectively. Metergoline is a high-affinity ligand for the h5-HT 7 receptor, with a K i of 16 nM. Metergoline is also a reversible neural Na + channels inhibitor. Metergoline is commonly used for the research of seasonal affective disorder, prolactin hormone regulation.

Application

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Product Information

• Catalog No.: HY-B1033
• CAS No.: 17692-51-2
• Molecular Formula: C25H29N3O2
• Molecular Weight: 403.52
• Purity: 99.94%
• Storage: Powder -20°C, 3 years ; In solvent -80°C, 6 months , -20°C, 1 month
• Solubility: ≥ 2.08 mg/mL (5.15 mM); Clear solution
• Availability: In-stock

Source

Original product source