AGN 193109

Overview

AGN 193109 is a retinoid analog, and acts as a specific and highly effective antagonist of retinoic acid receptors (RARs) , with K d s of 2 nM, 2 nM, and 3 nM for RARα , RARβ , and RARγ , respectively. AGN 193109 is a click chemistry reagent, it contains an Alkyne group and can undergo copper-catalyzed azide-alkyne cycloaddition (CuAAc) with molecules containing Azide groups. AGN 193109 is the antidote for retinoic acidosis, that ameliorates the skin and mucosal toxicity.

Application

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Product Information

• Catalog No.: HY-U00449
• CAS No.: 171746-21-7
• Molecular Formula: C28H24O2
• Molecular Weight: 392.49
• Purity: 99.80%
• Storage: Powder -20°C, 3 years ; In solvent -80°C, 2 years , -20°C, 1 year
• Solubility: ≥ 0.4 mg/mL (1.02 mM); Clear solution
• Availability: In-stock

Source

Original product source