(+)-JQ-1

Overview

(+)-JQ-1 is a potent and selective BET bromodomain inhibitor, IC50 values are 77 nM and 33 nM for inhibiting BRD4 (N-terminal) and BRD4 (C-terminal), respectively.

Application

Products > Drug Discovery > Inhibitor | Products > Drug Discovery > Inhibitor | Cancer | BET Bromodomain

Product Information

• Catalog No.: B0084-453787
• CAS No.: 1268524-70-4
• Molecular Formula: C₂₃H₂₅ClN₄O₂S
• Molecular Weight: 456.99
• Storage: Powder, -20°C, 3 years; 4°C, 2 years; In solvent, -80°C, 6 months; -20°C, 1 month
• Solubility: In DMSO: ≥ 45 mg/mL (98.47 mM) * "≥" means soluble, but saturation unknown.

Source

Original product source