A-366

Overview

A-366 is a peptide-competitive inhibitor of the G9a/GLP histone lysine methyltransferase (IC50 = 3.3 nM) and is approximately 1000-fold selective over other methyltransferases.

Application

Products > Drug Discovery > Inhibitor | Products > Drug Discovery > Inhibitor | Cancer | HMTase

Product Information

• Catalog No.: B2693-474604
• CAS No.: 1527503-11-2
• Molecular Formula: C19H27N3O2
• Molecular Weight: 329.44
• Storage: Store in a cool and dry place and at 0 - 4°C for short term (days to weeks) or -57°C for long term (months to years).
• Solubility: Soluble to 100 mM in 1eq. HCl and to 100 mM in DMSO

Source

Original product source