R547

Overview

R547 is a potent, selective and orally active ATP-competitive CDK inhibitor, with K i s of 2 nM, 3 nM and 1 nM for CDK1/cyclin B, CDK2/cyclin E and CDK4/cyclin D1, respectively.

Application

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Product Information

• Catalog No.: HY-10014
• CAS No.: 741713-40-6
• Molecular Formula: C18H21F2N5O4S
• Molecular Weight: 441.45
• Purity: 99.57%
• Storage: Powder -20°C, 3 years , 4°C, 2 years ; In solvent -80°C, 2 years , -20°C, 1 year
• Solubility: ≥ 2.5 mg/mL (5.66 mM); Clear solution
• Availability: In-stock

Source

Original product source