GSK484 hydrochloride

Overview

GSK484 hydrochloride is a selective and reversible peptidylarginine deiminase 4 ( PAD4 ) inhibitor. GSK484 hydrochloride demonstrates high affinity binding to PAD4 with IC 50 s of 50 nM in the absence of Calcium. In the presence of 2 mM Calcium, notably lower potency (250 nM) is observed.

Application

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Product Information

• Catalog No.: HY-100514
• CAS No.: 1652591-81-5
• Molecular Formula: C27H32ClN5O3
• Molecular Weight: 510.03
• Purity: 99.48%
• Storage: 4°C, stored under nitrogen, away from moisture * In solvent : -80°C, 1 year; -20°C, 6 months (stored under nitrogen, away from moisture)
• Solubility: ≥ 2.08 mg/mL (4.08 mM); Clear solution
• Availability: In-stock

Source

Original product source