Hydroxybupropion

Overview

Hydroxybupropion is the major active metabolite of Bupropion. Hydroxybupropion is metabolized by CYP2B6. Bupropion is an atypical antidepressant and smoking-cessation agent. Hydroxybupropion inhibits norepinephrine uptake with an IC 50 value of 1.7 μM. Hydroxybupropion is also a nACh receptor antagonist .

Application

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Product Information

• Catalog No.: HY-100637
• CAS No.: 92264-81-8
• Molecular Formula: C13H18ClNO2
• Molecular Weight: 255.74
• Purity: 99.91%
• Storage: Powder -20°C, 3 years , 4°C, 2 years ; In solvent -80°C, 6 months , -20°C, 1 month
• Solubility: ≥ 2.5 mg/mL (9.78 mM); Clear solution
• Availability: In-stock

Source

Original product source