GSK2193874

Overview

GSK2193874 is an orally active, potent, and selective TRPV4 antagonist with IC 50 s of 2 nM and 40 nM for rTRPV4 and hTRPV4 .

Application

Products | Products > Disease Areas > Neurological, Eye or Ear Disease | Products > Disease Areas > Blood or Cardio-cerebrovascular Disease | Products > Disease Areas > Pain | Products > Disease Areas > Cardiovascular Disease | Products > Signaling Pathways > Membrane Transporter/Ion Channel | Products > Signaling Pathways > Neuronal Signaling | Products > Research Areas > Cardiovascular Disease | Products > Signaling Pathways > TRP Channel

Product Information

• Catalog No.: HY-100720
• CAS No.: 1336960-13-4
• Molecular Formula: C37H38BrF3N4O
• Molecular Weight: 691.62
• Purity: 99.91%
• Storage: Powder -20°C, 3 years , 4°C, 2 years ; In solvent -80°C, 2 years , -20°C, 1 year
• Solubility: ≥ 2.08 mg/mL (3.01 mM); Clear solution
• Availability: In-stock

Source

Original product source