CHS-828

Overview

CHS-828 (GMX1778) is a competitive inhibitor of nicotinamide phosphoribosyltransferase ( NAMPT ) , with an IC 50 less than 25 nM. CHS-828 (GMX1778) exerts a cytotoxic effect by decreasing the cellular level of NAD + and exhibits a potent anticancer activity.

Application

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Product Information

• Catalog No.: HY-10079
• CAS No.: 200484-11-3
• Molecular Formula: C19H22ClN5O
• Molecular Weight: 371.86
• Purity: 99.28%
• Storage: Powder -20°C, 3 years , 4°C, 2 years ; In solvent -80°C, 2 years , -20°C, 1 year
• Solubility: ≥ 2.5 mg/mL (6.72 mM); Clear solution
• Availability: In-stock

Source

Original product source