Teglarinad chloride

Overview

Teglarinad chloride (GMX1777) is a proagent of GMX1778 (a nicotinamide phosphoribosyl transferase inhibitor). Teglarinad chloride exhibits antitumor activity in mice can be attributed to inhibition of NAMPT . Teglarinad chloride also enhances radiation efficacy, mediated by interference with DNA repair and antiangiogenesis.

Application

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Product Information

• Catalog No.: HY-10080
• CAS No.: 432037-57-5
• Molecular Formula: C30H43Cl2N5O8
• Molecular Weight: 672.60
• Purity: 99.67%
• Storage: -20°C, sealed storage, away from moisture * In solvent : -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture)
• Solubility: ≥ 3.75 mg/mL (5.58 mM); Clear solution
• Availability: In-stock

Source

Original product source