GKT136901 hydrochloride

Overview

GKT136901 hydrochloride is a potent, selective and orally active inhibitor of NADPH oxidase (NOX1/4) , with K i s of 160 and 165 nM, respectively. GKT136901 hydrochloride is also a selective and direct scavenger of peroxynitrite. GKT136901 hydrochloride can be used for the research of diabetic nephropathy, stroke, and neurodegeneration. GKT136901 hydrochloride also has anti-inflammatory activity.

Application

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Product Information

• Catalog No.: HY-101499A
• CAS No.: 1254507-01-1
• Molecular Formula: C19H16Cl2N4O2
• Molecular Weight: 403.26
• Purity: 99.59%
• Storage: 4°C, sealed storage, away from moisture * In solvent : -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture)
• Solubility: ≥ 2.08 mg/mL (5.16 mM); Clear solution
• Availability: In-stock

Source

Original product source