NNC-711

Overview

NNC-711 (NO-711 hydrochloride) is a potent and selective inhibitor of GAT-1 (GABA transporter 1) with IC 50 values of 0.04, 0.38, 171, 1700, 349, 622 μM for human GAT-1, rat GAT-1, rGAT-2, hGAT-3, rGAT-3, hBGT-3, respectively. NNC-711 has anticonvulsant and analgesic effect in vivo and exhibits cognition-enhancing activity.

Application

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Product Information

• Catalog No.: HY-103506
• CAS No.: 145645-62-1
• Molecular Formula: C21H23ClN2O3
• Molecular Weight: 386.87
• Purity: 99.76%
• Storage: -20°C, sealed storage, away from moisture * In solvent : -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture)
• Solubility: ≥ 2.5 mg/mL (6.46 mM); Clear solution
• Availability: In-stock

Source

Original product source