Velusetrag hydrochloride

Overview

Velusetrag (TD-5108) hydrochloride is an orally active, potent and selective agonist of serotonin 5-HT 4 receptor (5-HT 4 R) , with a pK i of 7.7. Velusetrag hydrochloride exhibits no affinity (K i >10 μM) for 5-HT 2A and 5-HT 2B receptors. Velusetrag hydrochloride can be used for the research of gastrointestinal diseases and Parkinson's disease.

Application

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Product Information

• Catalog No.: HY-10457A
• CAS No.: 866933-51-9
• Molecular Formula: C25H37ClN4O5S
• Molecular Weight: 541.10
• Purity: 98.95%
• Storage: 4°C, sealed storage, away from moisture * In solvent : -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture)
• Solubility: ≥ 5.5 mg/mL (10.16 mM); Clear solution
• Availability: In-stock

Source

Original product source