CCR2 antagonist 4

Overview

CCR2 antagonist 4 (Teijin compound 1) is a potent and specific CCR2 antagonist, with IC 50 s of 180 nM for CCR2b. CCR2 antagonist 4 potently inhibits MCP-1-induced chemotaxis with an IC 50 of 24 nM.

Application

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Product Information

• Catalog No.: HY-108323
• CAS No.: 226226-39-7
• Molecular Formula: C21H21ClF3N3O2
• Molecular Weight: 439.86
• Purity: 100.0%
• Storage: Powder -20°C, 3 years , 4°C, 2 years ; In solvent -80°C, 6 months , -20°C, 1 month
• Solubility: ≥ 2.5 mg/mL (5.68 mM); Clear solution
• Availability: In-stock

Source

Original product source