WHI-P258

Overview

WHI-P258, a quinazoline compound, binds to the active site of JAK3 with an estimated K i of 72 µM. WHI-P258 does not inhibit JAK3 and does not affect the thrombin-induced aggregation of platelets even at 100 μM.

Application

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Product Information

• Catalog No.: HY-108419
• CAS No.: 21561-09-1
• Molecular Formula: C16H15N3O2
• Molecular Weight: 281.31
• Purity: 99.91%
• Storage: Powder -20°C, 3 years , 4°C, 2 years ; In solvent -80°C, 2 years , -20°C, 1 year
• Solubility: ≥ 2.25 mg/mL (8.00 mM); Clear solution
• Availability: In-stock

Source

Original product source