GNE-049

Overview

GNE-049 is a highly potent and selective CBP inhibitor with an IC 50 of 1.1 nM in TR-FRET assay. GNE-049 also inhibits BRET and BRD4(1) with IC 50 s of 12 nM and 4200 nM, respectively.

Application

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Product Information

• Catalog No.: HY-108435
• CAS No.: 1936421-41-8
• Molecular Formula: C27H32F2N6O2
• Molecular Weight: 510.58
• Purity: 99.74%
• Storage: -20°C, stored under nitrogen * In solvent : -80°C, 6 months; -20°C, 1 month (stored under nitrogen)
• Availability: In-stock

Source

Original product source