VU0650786

Overview

VU0650786 is a potent and selective CNS penetrant negative allosteric modulator of metabotropic glutamate receptor subtype 3 (mGlu3 NAM) , with an IC 50 of 392 nM. VU0650786 has antidepressant and anxiolytic activity in rodents.

Application

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Product Information

• Catalog No.: HY-108710
• CAS No.: 1809085-30-0
• Molecular Formula: C18H15ClFN5O2
• Molecular Weight: 387.80
• Purity: 99.55%
• Storage: Powder -20°C, 3 years , 4°C, 2 years ; In solvent -80°C, 6 months , -20°C, 1 month
• Solubility: ≥ 2.08 mg/mL (5.36 mM); Clear solution
• Availability: In-stock

Source

Original product source